AP-238

AP-238

AP-238 is a new opioid drug 5 times more effective than morphine, it is an excellent analgesic, it is very popular in Asia for the treatment of cancer patients. AP-238 is a µ-opioid receptor (MOR) agonist with a relatively low affinity for the δ-opioid receptor and κ-opioid receptor. When used regularly, AP-238 can quickly develop drug tolerance and addiction.

 

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Description

Synonyms

​2,6-dimethyl Propionyl AP-237
Technical Information
Formal Name
1-[2,6-dimethyl-4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]-1-propanone, monohydrochloride
CAS Number
2749171-05-7
Molecular Formula
C18H26N2O • HCl
Formula Weight
322.9
Purity
≥98%
Formulation
(Request formulation change)
A crystalline solid
Solubility
(Learn about Variance in Solubility)
DMF: 10 mg/ml
DMSO: 15 mg/ml
Ethanol: 30 mg/ml
PBS (pH 7.2): 10 mg/ml
λmax
254 nm
SMILES
CCC(N1C(C)CN(C/C=C/C2=CC=CC=C2)CC1C)=O.Cl
InChi Code
InChI=1S/C18H26N2O.ClH/c1-4-18(21)20-15(2)13-19(14-16(20)3)12-8-11-17-9-6-5-7-10-17;/h5-11,15-16H,4,12-14H2,1-3H3;1H/b11-8+;
InChi Key
MKVRJEWKXNVTIF-YGCVIUNWSA-N

Shipping & Storage Information

Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 5 years