N-Desmethyl-loperamide

Loperamide is a synthetic opiate that efficiently and selectively activates the μ opioid receptors Ki = 0.16 nM, exclusively at the periphery. N-Desmethyl-loperamide (dLop) is the main metabolite of loperamide. dLop is a substrate of an ATP-dependent outflow conveyor, P-glycoprotein. As a result, both the initial compound and the mapping of metabolites, limited by passage through the blood, can be analyzed by various methods.

• N-Desmethyl-loperamide 10g 139 € Order form
  
• N-Desmethyl-loperamide 100g 690 € Order form
  
• N-Desmethyl-loperamide 500g 1490 € Order form
  
• N-Desmethyl-loperamide 1 kg 1990 € Order form