LY2183240

LY2183240

LY2183240 and all other synthetic product of cannabinoids sold on this website are intended for a research and court affidavits. The research the chemical new design drug called by LY2183240 with the obvious physiological and influencing mentality effects also has a molecular formula C17H17N5O. The weight of a formula has a cost of 307.4 g / molecular masses.

LY2183240 10g 79€ Order form

LY2183240 50g 249€ Order form

LY2183240 100g 399€ Order form

LY2183240 500g 1190€ Order form

LY2183240 1kg 1690€ Order form

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Description

Buy bulk LY2183240 Online

LY2183240 is a highly potent blocker of anandamide uptake (IC50= 270 pM; Ki=540 nM). LY2183240 is a potent, covalent inhibitor of the endocannabinoid-degrading enzyme fatty acid amide hydrolase (FAAH) with an IC50 of 12.4 nM. LY2183240 inactivates FAAH by carbamylation of the enzyme’s serine nucleophile. LY2183240 also inhibits several other brain serine hydrolases with IC50s of 5.3, 0.09, 8.2 nM for MAG lipase, bh6 and KIAA1363, respectively .

LY-2183240 is a potent, covalent inhibitor of the EC-degrading enzyme fatty acid amide hydrolase (FAAH). LY-2183240 disrupts the cellular uptake of the lipid endocannabinoid (EC) anandamide and promote analgesia in vivo. LY-2183240 is also an inhibitor of monoacylgylcerol lipase (MGL).

Technical Information
Formal Name
5-([1,1′-biphenyl]-4-ylmethyl)-N,N-dimethyl-1H-tetrazole-1-carboxamide
CAS Number
874902-19-9
Molecular Formula
C17H17N5O
Formula Weight
307.4
Purity
≥98%
Formulation
(Request formulation change)
A crystalline solid
Solubility
(Learn about Variance in Solubility)
DMF: 3 mg/ml
DMSO: 2 mg/ml
Ethanol: 10 mg/ml
Ethanol:PBS(pH 7.2) (1:5): 0.1 mg/ml
λmax
253 nm
SMILES
O=C(N(C)C)N1N=NN=C1CC2=CC=C(C3=CC=CC=C3)C=C2
InChi Code
InChI=1S/C17H17N5O/c1-21(2)17(23)22-16(18-19-20-22)12-13-8-10-15(11-9-13)14-6-4-3-5-7-14/h3-11H,12H2,1-2H3
InChi Key
GZNIYOXWFCDBBJ-UHFFFAOYSA-N

Shipping & Storage Information

Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 2 years